Oxacillin

Dose Adult

Mild to moderate infections: 250–500 mg orally every 6 hours.

Severe MSSA infections: 1–2 g IV every 4–6 hours.

Endocarditis/Osteomyelitis: Up to 12 g/day IV in divided doses.

Dose Paeds

50–100 mg/kg/day in divided doses every 6 hours.

Severe infections: Up to 200 mg/kg/day IV in divided doses.

Oxacillin Brands

BrandManufacturerDistributorStrengthPackagingFormulationPrice
BactocillPfizerVarious500 mgVialPowder for InjectionKES POR
Oxacillin SodiumGenericVarious1 gVialPowder for InjectionKES POR
Oxacillin SodiumGenericVarious2 gVialPowder for InjectionKES POR

Combinations

Usually used alone. May be combined clinically with aminoglycosides for selected severe infections (administer separately).

Oxacillin More action
IndicationsMethicillin-sensitive Staphylococcus aureus (MSSA) infections, cellulitis, osteomyelitis, septic arthritis, endocarditis, pneumonia, bacteraemia and skin/soft tissue infections.
PrecautionsHistory of penicillin allergy, hepatic impairment, renal impairment, prolonged therapy, monitor liver function and blood counts.
ContraindicationsKnown hypersensitivity to oxacillin, penicillins or other beta-lactam antibiotics.
Pregnancy/LactationPregnancy Category B. Generally considered safe during pregnancy and breastfeeding when clinically indicated.
Adverse reactionRash, urticaria, anaphylaxis, nausea, diarrhoea, hepatitis, neutropenia, interstitial nephritis, phlebitis and superinfection.
PolypharmacyMay interact with warfarin, methotrexate and probenecid. Avoid mixing in the same IV line with aminoglycosides. Monitor anticoagulant response when co-administered.
Drug CategoryDRUGS ACTING ON INFECTIONS
Drug Sub-CategoryPenicillinase-resistant Penicillins