Rizatriptan

Dosage ; Single doses of 5 and 10 mg.

Redosing: Doses should be separated by at least 2 hours, no more than 30mg should be taken in any 24-hour period.

The safety of treating, on average,

more than four headaches in a 30-day period has not been established.

Rizatriptan Brands

Brand Name Manufacturer Name Distributor Drug Strength Packaging Formulation Formulation Strength Price
Imigran

NB; Not Imigram

GlaxoSmithkline GlaxoSmithKline 100mg 6 Tablet per tablet KES 6,691.60
Rizat Cipla Ltd. Lords Healthcare Ltd. 10mg 4 Tablet per tablet KES 1,035
Rizact Cipla Ltd. Surgipharm Ltd 10mg 4 Tablet per tablet KES 1,200.00

Rizatriptan More info

Mode Of Action

Serotonin (5HTI) agonist

Drug Indication Migraine (acute), cluster headache
Precautions Renal, hepatic, neurological and CV disorders, epilepsy, sulphonamide sensitivity
Contra-Indications Uncontrolled hypertension, SC use in patients with ischaemic heart disease, concomitant use with ergotamine preparations, management of hemiplegic or basilar migraine, IV use.
Side Effects Burning sensation, tingling, warm/hot sensation, visual disturbances, nasal
Dosage Single doses of 5 and 10 mg. Redosing: Doses should be separated by at least 2 hours, no more than 30mg should be taken in any 24-hour period. The safety of treating, on average, more than four headaches in a 30-day period has not been established.
Special Information It is structurally as well as pharmacologically related to serotonin, (5-hydroxytryptamine, 5HT) differing structurally from serotonin mainly by the substitution of methane sulfonamide for the alcohol group on the indication sole ring.
Drug Category DRUGS ACTING ON CNS
Drug Sub-Category Anti-migraine drugs

Dosing: Adult

Note: In patients with risk factors for coronary artery disease, following adequate evaluation to establish the absence of coronary artery disease, the initial dose should be administered in a setting where response may be evaluated (physician's office or similarly staffed setting). ECG monitoring may be considered.

Migraine: Oral: 5-10 mg, repeat after 2 hours if significant relief is not attained; maximum: 30 mg in a 24-hour period (use 5 mg dose in patients receiving propranolol with a maximum of 15 mg in 24 hours)

Note: For orally-disintegrating tablets (Maxalt-MLT®): Patient should be instructed to place tablet on tongue and allow to dissolve. Dissolved tablet will be swallowed with saliva.

Dosing: Geriatric

Refer to adult dosing